Prostate cancer

45 imaging agents and 64 therapeutic agents reported for this indication. Stage reflects how far each has been taken, not what is available in any given country.

Imaging

Agent	Isotope	Stage	Runs
[68Ga]Ga-PSMA-11 paired with [177Lu]Lu-PSMA-617	Ga-68	Approved	56
[18F]PSMA-1007 paired with [177Lu]Lu-PSMA-617	F-18	Clinical research	11
[18F]fluoroethylcholine	F-18	—	11
[68Ga]Ga-PSMA-617	Ga-68	Clinical research	9
[68Ga]Ga-RM2 paired with [111In]In-RM2	Ga-68	Clinical research	7
[11C]choline	C-11	Approved	6
[18F]DCFPyL paired with [177Lu]Lu-PSMA-617	F-18	Approved	5
[68Ga]Ga-PSMA-I&T paired with [177Lu]Lu-PSMA-I&T	Ga-68	—	5
[18F]rhPSMA-7 paired with [177Lu]Lu-rhPSMA-7	F-18	Clinical research	4
[99mTc]Tc-PSMA-I&S	Tc-99m	—	4
[111In]In-RM2 paired with [68Ga]Ga-RM2	In-111	Research	2
[18F]AlF-P16-093	F-18	—	2
[18F]FDHT	F-18	—	2
[18F]F-PSMA-617-NODA	F-18	—	2
[18F]F-PSMA-617-RESCA	F-18	—	2
[18F]JK-PSMA-7	F-18	—	2
[11C]PD153035	C-11	Clinical research	1
[11C]YM155	C-11	—	1
[18F]FACBC	F-18	Approved	1
[18F]FCH	F-18	—	1
[68Ga]Ga-FAPI-74	Ga-68	—	1
[68Ga]Ga-NOTA-BBN2	Ga-68	Preclinical	1
[99mTc]Tc-N4-PSMA-12	Tc-99m	Preclinical	1
[99mTc]Tc-TcO2	Tc-99m	Preclinical	1
[68Ga]PKB2	Ga-68	Reported once	1
[68Ga]PKB3	Ga-68	Reported once	1
[86Y]pepa-pic2-C-Hex-KuE	Y-86	Reported once	1
[68Ga]PSMA-1-DOTA paired with [177Lu]Lu-PSMA-1-DOTA	Ga-68	Clinical research	1
[68Ga]LW02060 paired with [177Lu]Lu-LW02060	Ga-68	Reported once	1
[68Ga]LW02080 paired with [177Lu]Lu-LW02080	Ga-68	Reported once	1
[68Ga]HTK03177	Ga-68	Preclinical	1
[68Ga]HTK03187	Ga-68	Reported once	1
[18F]AlF-3p-C-NETA-ePSMA-16	F-18	Preclinical	1
[68Ga]HTK03161	Ga-68	Reported once	1
[68Ga]HTK03149 paired with [177Lu]Lu-HTK03149	Ga-68	Reported once	1
[68Ga]HTK03189B	Ga-68	Reported once	1
[89Zr]hu5A10	Zr-89	Preclinical	1
[68Ga]177-AAZTA5-PSMA-617 paired with [177Lu]Lu-177-AAZTA5-PSMA-617	Ga-68	Preclinical	1
[44Sc]177-AAZTA5-PSMA-617	Sc-44	Preclinical	1
[111In]In-PSMA-617 paired with [177Lu]Lu-PSMA-617	In-111	Research
[18F]FSO3-PSMA	F-18	Research
[18F]ef5	F-18	—
[68Ga]Ga-P16-093	Ga-68	Clinical research
[99mTc]Tc-N4-Bombesin	Tc-99m	Preclinical
[68Ga]TacsBOMB2	Ga-68	Preclinical

Therapy

Agent	Isotope	Stage	Runs
[177Lu]Lu-PSMA-617 paired with [68Ga]Ga-PSMA-11	Lu-177	Approved	35
[177Lu]Lu-PSMA-I&T paired with [68Ga]Ga-PSMA-I&T	Lu-177	Clinical research	20
[225Ac]Ac-PSMA-617 paired with [111In]In-PSMA-617	Ac-225	Clinical research	5
[225Ac]Ac-PSMA-I&T paired with [68Ga]Ga-PSMA-I&T	Ac-225	Clinical research	4
[225Ac]Ac-DOTA-YS5	Ac-225	Preclinical	4
[153Sm]Sm-EDTMP	Sm-153	Approved	3
[223Ra]Ra-RaCl2	Ra-223	Approved	3
[177Lu]Lu-AMTG	Lu-177	Clinical research	3
[177Lu]Lu-PSMA-ALB-56	Lu-177	—	3
[177Lu]Lu-AMBA	Lu-177	—	3
[225Ac]Ac-Macropa-PEG4-YS5	Ac-225	—	3
[177Lu]Lu-CTT2001	Lu-177	Clinical research	2
[177Lu]Lu-P17-087	Lu-177	Clinical research	2
[177Lu]Lu-P17-088	Lu-177	Clinical research	2
[212Pb]Pb-PSMA-617 paired with [111In]In-PSMA-617	Pb-212	—	2
[177Lu]Lu-rhPSMA-7 paired with [18F]rhPSMA-7	Lu-177	—	2
[211At]At-PSMA-5	At-211	Preclinical	2
[177Lu]Lu-Ibu-DAB-PSMA	Lu-177	Preclinical	2
[212Pb]Pb-AB001	Pb-212	—	2
[177Lu]Lu-PSMA-10	Lu-177	Preclinical	1
[47Sc]Sc-PSMA-617 paired with [111In]In-PSMA-617	Sc-47	Preclinical	1
[161Tb]Tb-RM2 paired with [68Ga]Ga-RM2	Tb-161	Preclinical	1
[161Tb]Tb-PSMA-I&T paired with [68Ga]Ga-PSMA-I&T	Tb-161	Clinical research	1
[188Re]Re-188-HEDP	Re-188	Clinical research	1
[177Lu]Lu-LuCl3	Lu-177	—	1
[90Y]Y-90-NM600	Y-90	Preclinical	1
[225Ac]Ac-90-NM600	Ac-225	Preclinical	1
[177Lu]Lu-NeoBOMB1	Lu-177	—	1
[161Tb]Tb-AMTG	Tb-161	Preclinical	1
[177Lu]Lu-NeoB	Lu-177	Clinical research	1
[225Ac]Ac-mcp-TDI-Y-010	Ac-225	Reported once	1
[177Lu]Lu-pepa-pic2-C-Hex-KuE	Lu-177	Reported once	1
[161Tb]Tb-pepa-pic2-C-Hex-KuE	Tb-161	Preclinical	1
[177Lu]Lu-PSMA-1-DOTA paired with [68Ga]PSMA-1-DOTA	Lu-177	Clinical research	1
[177Lu]Lu-LW01110	Lu-177	Preclinical	1
[177Lu]Lu-LW01142	Lu-177	Reported once	1
[212Pb]Pb-DOTAM-GRPR1	Pb-212	Preclinical	1
[211At]At-L3-Lu	At-211	Reported once	1
[177Lu]Lu-PEG-(DOTA)1	Lu-177	Preclinical	1
[177Lu]Lu-PEG-(DOTA)1(ACUPA)3	Lu-177	Reported once	1
[177Lu]Lu-HTK03170	Lu-177	Preclinical	1
[111In]3p-C-NETA-ePSMA-16	In-111	Preclinical	1
[177Lu]Lu-3p-C-NETA-ePSMA-16	Lu-177	Preclinical	1
[213Bi]Bi-3p-C-NETA-ePSMA-16	Bi-213	Preclinical	1
[177Lu]Lu-HTK03149 paired with [68Ga]HTK03149	Lu-177	Reported once	1
[111In]BQ7859	In-111	Reported once	1
[90Y]Y-hu5A10	Y-90	Preclinical	1
[225Ac]Ac-hu5A10	Ac-225	Reported once	1
[177Lu]Lu-177-AAZTA5-PSMA-617 paired with [68Ga]177-AAZTA5-PSMA-617	Lu-177	Reported once	1
[125I]I-BO530	I-125	Reported once	1
[131I]PSMA-769	I-131	Reported once	1
[131I]PSMA-769-d-tyrosine	I-131	Preclinical	1
[177Lu]Lu-rhPSMA-10	Lu-177	Clinical research
[161Tb]Tb-PSMA-617 paired with [111In]In-PSMA-617	Tb-161	Clinical research
[213Bi]Bi-PSMA-617 paired with [111In]In-PSMA-617	Bi-213	—
[177Lu]Lu-J591	Lu-177	Clinical research
[225Ac]Ac-J591	Ac-225	Clinical research
[177Lu]Lu-SibuDAB	Lu-177	—
[225Ac]Ac-SibuDAB	Ac-225	Clinical research
[177Lu]Lu-PSMA-617-treated	Lu-177	Clinical research
[177Lu]Lu-LNC1011	Lu-177	Clinical research
[211At]At-astatinated	At-211	—
[177Lu]Lu-vipivotide	Lu-177	Approved
[225Ac]Ac-225-DOTA-J591	Ac-225	Clinical research

Other entries

Agent	Isotope	Stage	Runs
[57Co]Co-NOTA-PEG2-RM26	Co-57	Preclinical	2
[68Ga]Ga-DATA5m.SA.FAPi	Ga-68	Clinical research	1
[64Cu]CuCl2	Cu-64	Clinical research	1
[90Y]Y-DOTA-AR	Y-90	Preclinical	1
[225Ac]Ac-PSMA-RLT	Ac-225	—
[64Cu]Cu-AuNPs	Cu-64	—

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