Tracers / [111In]3p-C-NETA-ePSMA-16

[111In]3p-C-NETA-ePSMA-16

Also written as [In-111]In-3p-C-NETA-ePSMA-16
Radionuclide
In-111 t½ 4031.6 min
Modality
Therapy
Production route
Stage
Reported once
Syntheses indexed
1

What it is

Compound class
PSMA-targeting NETA-based bifunctional chelator conjugate (PSMA-targeting radiotheranostic agent)
Target / mechanism
PSMA (prostate-specific membrane antigen) PMID 37375829
Clinical application
Theranostic pair

Regulatory status

FDA
EMA (centralised)
Other approvals
Brand names

Clinical use

Typical injected activity
Uptake time

Reported in the literature. Not a dosing recommendation.

Published syntheses

ModuleCassettePurificationYield %RCP %Precursor / supplierSource
Manual synthesis99.7 ± 0.2%>99%3p-C-NETA-ePSMA-1637375829
2023 Pharmaceuticals (Basel)
Radiolabeling with 111In afforded quantitative radiochemical yield (RCY) (99.7 ± 0.2%, n = 5) in mild conditions (rt, 5 min) — Radiolabeling with 111In afforded quantitative radiochemical yield (RCY) (99.7 ± 0.2%, n = 5)

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Notes

Added at stage 22: promoted from 'Reported once' (single-article, no diagnostic pair at discovery) because a full-text synthesis with extracted data exists in parsed-therapy.xlsx -- PMID(s): 37375829. Target/mechanism, clinical application, indications, approval and precursor fields still need per-agent research and are intentionally left empty. Compound class inferred from precursor name (not stated outright) -- PMID 37375829: '3p-C-NETA-ePSMA-16 (1 nmol) dissolved in H2O was added to the solution'.