Tracers / [213Bi]Bi-PSMA-617

[213Bi]Bi-PSMA-617

Also written as PSMA-617; Pluvicto
Radionuclide
Bi-213 t½ 45.6 min
Modality
Therapy
Production route
Stage
Syntheses indexed
1

What it is

Compound class
PSMA-targeting small molecule (urea-based PSMA ligand)
Target / mechanism
Prostate-specific membrane antigen (PSMA) PMID 28891033
Clinical application
Targeted alpha therapy of metastatic castration-resistant prostate cancer (dosimetry estimate) PMID 28891033
Theranostic pair
<a href="/tracers/in111-psma617/">in111-psma617</a>

Regulatory status

FDA
EMA (centralised)
Other approvals
Brand names

Clinical use

Typical injected activity
Uptake time

Reported in the literature. Not a dosing recommendation.

Published syntheses

ModuleCassettePurificationYield %RCP %Precursor / supplierSource
28891033
2018 Eur J Nucl Med Mol Imaging

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Notes

Added at stage 21 from therapy-discovered.xlsx (bulk PubMed search by isotope/therapy-type/known-agent, not individually researched yet) -- 1 articles found. Target/mechanism, clinical application, indications, approval and precursor fields still need per-agent research and are intentionally left empty. Diagnostic pair signal at discovery: YES - Ga-68, In-111.