By indication / Dosimetry and biodistribution studies

Dosimetry and biodistribution studies

32 imaging agents and 41 therapeutic agents reported for this indication. Stage reflects how far each has been taken, not what is available in any given country.

Imaging

AgentIsotopeStageRuns
[68Ga]Ga-PSMA-617Ga-68Clinical research9
[18F]rhPSMA-7
paired with [177Lu]Lu-rhPSMA-7
F-18Clinical research4
[18F]AmBF3-TATEF-18Preclinical3
[18F]PBR111F-18—3
[111In]In-RM2
paired with [68Ga]Ga-RM2
In-111Research2
[18F]FEDAA1106F-18Clinical research2
[18F]PBR102F-18Preclinical2
10-[11C]methoxy-20(S)-camptothecinC-11Preclinical1
[11C]PD153035C-11Clinical research1
[18F]ApaScanF-18Preclinical1
[18F]BTK-1F-18Preclinical1
[18F]FB-A20FMDV2F-18Preclinical1
[18F]FBEM-Cys-H4F-18Preclinical1
[18F]MEL050F-18Clinical research1
[68Ga]Ga-BOT5035Ga-68Clinical research1
[111In]DOTA-MSC3In-111Preclinical1
[111In]BCY18469In-111Preclinical1
[68Ga]NOTA-MI-exendin-4Ga-68Preclinical1
[68Ga]HTK03149
paired with [177Lu]Lu-HTK03149
Ga-68Reported once1
[89Zr]hu5A10Zr-89Preclinical1
[99mTc]Tc(CO)3-ADAPT6Tc-99mPreclinical1
[111In]In-PSMA-617
paired with [177Lu]Lu-PSMA-617
In-111Research
[11C]KIn83C-11—
[11C]Me-NB1C-11Clinical research
[18F]AF78F-18Clinical research
[18F]fiauF-18Clinical research
[18F]fluoro-3-(2(S)-azetidinylmethoxy)pyridineF-18—
[18F]fluorophenylalanineF-18Clinical research
[18F]L-GlutamicF-18Clinical research
[68Ga]Ga-oxineGa-68Clinical research
[68Ga]Ga-P16-093Ga-68Clinical research
[89Zr]vMET1-Fc
paired with [177Lu]Lu-vMET1-Fc
Zr-89Preclinical

Therapy

AgentIsotopeStageRuns
[177Lu]Lu-DOTA-TOC
paired with [68Ga]Ga-DOTA-TOC
Lu-177—11
[177Lu]Lu-DOTA-MGS5Lu-177Clinical research8
[225Ac]Ac-DOTATATE
paired with [68Ga]Ga-DOTATATE
Ac-225Clinical research4
[225Ac]Ac-PSMA-I&T
paired with [68Ga]Ga-PSMA-I&T
Ac-225Clinical research4
[161Tb]Tb-crownTb-161Preclinical4
[177Lu]Lu-PSMA-ALB-56Lu-177—3
[90Y]Y-L4-Lipo/Y-90Preclinical3
[161Tb]Tb-DOTA-LM3Tb-161Clinical research2
[188Re]Re-MAG3Re-188—2
[177Lu]Lu-GeminiLu-177—2
[177Lu]Lu-FAP-2286
paired with [68Ga]Ga-FAP-2286
Lu-177Clinical research1
[177Lu]Lu-NeoBLu-177Clinical research1
[177Lu]Lu-DOTA-RituximabLu-177—1
[188Re]Re-tricarbonyl(cyclopentadienylcarbonate)rheniumRe-188Preclinical1
[177Lu]Lu-CHX-A''-DTPA-F8Lu-177Reported once1
[225Ac]Ac-3p-C-DEPA-TFP-PEG4-trastuzumabAc-225Preclinical1
[177Lu]Lu-LW01110Lu-177Preclinical1
[177Lu]Lu-LW01142Lu-177Reported once1
[177Lu]Lu-DOTA-Affiline-22Lu-177Preclinical1
[225Ac]Ac-Macropa-N4MU01Ac-225Reported once1
[212Pb]Pb-DOTAM-GRPR1Pb-212Preclinical1
[177Lu]Lu-DOTA-MI-exendin-4Lu-177Reported once1
[125I]NaIO3I-125Reported once1
[177Lu]Lu-rhPSMA-10Lu-177Clinical research
[213Bi]Bi-DOTA-TOC
paired with [68Ga]Ga-DOTA-TOC
Bi-213Clinical research
[161Tb]Tb-PSMA-617
paired with [111In]In-PSMA-617
Tb-161Clinical research
[213Bi]Bi-PSMA-617
paired with [111In]In-PSMA-617
Bi-213—
[177Lu]Lu-J591Lu-177Clinical research
[177Lu]Lu-SibuDABLu-177—
[225Ac]Ac-SibuDABAc-225Clinical research
[131I]I-131-Lym-1I-131—
[153Sm]Sm-BPAMD
paired with [68Ga]Ga-BPAMD
Sm-153Preclinical
[177Lu]Lu-LNC1011Lu-177Clinical research
[166Ho]Ho-166-PLLAHo-166—
[90Y]Y-microsphereY-90Approved
[177Lu]Lu-177-OncoFAP-23Lu-177Preclinical
[90Y]Y-anti-CD66Y-90—
[177Lu]Lu-177-OPS201Lu-177Preclinical
[188Re]Re-CpTR-COOHRe-188—
[177Lu]Lu-EvansLu-177Clinical research
[177Lu]Lu-DOTA-EB-TATELu-177—

Other entries

AgentIsotopeStageRuns
[111In]In-minigastrinIn-111—2
[111In]In-exendinIn-111—2
[125I]CPCR4.3I-125Preclinical1
[64Cu]CuCl2Cu-64Clinical research1
[90Y]Y-DOTA-ARY-90Preclinical1
[111In-DTPA]MG0In-111—1
[166Ho]Ho-DTPAHo-166Preclinical
[131I]I-omburtamabI-131Clinical research
[225Ac]Ac-HuM195Ac-225Preclinical
[188Re]Re-LiposomePreclinical
[11C]3-MeO-4-APC-11Preclinical
[212Pb]Pb-VMT-alpha-NETPb-212Clinical research
[111In]In-labeled NZ-16In-111Preclinical
[111In]In-DOTA-IgGPreclinical
[188Re]Re-IBARe-188—
[99mTc]Tc-BMEDA liposomesTc-99m—
[188Re]Re-C1P5Re-188Preclinical
[67Cu]Cu-TCPPCu-67—

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