Tracers / [177Lu]Lu-rhPSMA-7

[177Lu]Lu-rhPSMA-7

Also written as [Lu-177]Lu-rhPSMA-7; rhPSMA-7.3
Radionuclide
Lu-177 t½ 9584.6 min
Modality
Therapy
Production route
Stage
Syntheses indexed
2

What it is

Compound class
PSMA-targeted radiohybrid (rh) ligand
Target / mechanism
Prostate-specific membrane antigen (PSMA) PMID 35086894
Clinical application
Endoradiotherapy (radioligand therapy) of prostate cancer PMID 35086894
Theranostic pair
<a href="/tracers/f18-rhpsma7/">f18-rhpsma7</a>

Regulatory status

FDA
EMA (centralised)
Other approvals
Brand names

Clinical use

Typical injected activity
Uptake time

Reported in the literature. Not a dosing recommendation.

Published syntheses

ModuleCassettePurificationYield %RCP %Precursor / supplierSource
>95%rhPSMA-7.336145382
2022 Pharmaceuticals (Basel)
Manual synthesis>95%rhPSMA-7.3 precursor35086894
2022 J Nucl Med
177Lu labeling of PSMA ligands according to standard manual procedures resulted in a radiochemical purity of more than 95%

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Notes

Added at stage 21 from therapy-discovered.xlsx (bulk PubMed search by isotope/therapy-type/known-agent, not individually researched yet) -- 1 articles found. Target/mechanism, clinical application, indications, approval and precursor fields still need per-agent research and are intentionally left empty. Diagnostic pair signal at discovery: YES - F-18.