By indication / PSMA-directed radioligand therapy

PSMA-directed radioligand therapy

1 imaging agents and 28 therapeutic agents reported for this indication. Stage reflects how far each has been taken, not what is available in any given country.

Imaging

AgentIsotopeStageRuns
[68Ga]HTK03149
paired with [177Lu]Lu-HTK03149
Ga-68Reported once1

Therapy

AgentIsotopeStageRuns
[177Lu]Lu-PSMA-617
paired with [68Ga]Ga-PSMA-11
Lu-177Approved35
[177Lu]Lu-PSMA-I&T
paired with [68Ga]Ga-PSMA-I&T
Lu-177Clinical research20
[225Ac]Ac-PSMA-617
paired with [111In]In-PSMA-617
Ac-225Clinical research5
[225Ac]Ac-PSMA-I&T
paired with [68Ga]Ga-PSMA-I&T
Ac-225Clinical research4
[177Lu]Lu-PSMA-ALB-56Lu-177—3
[177Lu]Lu-P17-087Lu-177Clinical research2
[177Lu]Lu-P17-088Lu-177Clinical research2
[177Lu]Lu-rhPSMA-7
paired with [18F]rhPSMA-7
Lu-177—2
[211At]At-PSMA-5At-211Preclinical2
[177Lu]Lu-Ibu-DAB-PSMALu-177Preclinical2
[212Pb]Pb-AB001Pb-212—2
[161Tb]Tb-PSMA-I&T
paired with [68Ga]Ga-PSMA-I&T
Tb-161Clinical research1
[177Lu]Lu-PSMA-1-DOTA
paired with [68Ga]PSMA-1-DOTA
Lu-177Clinical research1
[177Lu]Lu-HTK03170Lu-177Preclinical1
[177Lu]Lu-HTK03149
paired with [68Ga]HTK03149
Lu-177Reported once1
[177Lu]Lu-rhPSMA-10Lu-177Clinical research
[161Tb]Tb-PSMA-617
paired with [111In]In-PSMA-617
Tb-161Clinical research
[213Bi]Bi-PSMA-617
paired with [111In]In-PSMA-617
Bi-213—
[177Lu]Lu-J591Lu-177Clinical research
[225Ac]Ac-J591Ac-225Clinical research
[177Lu]Lu-SibuDABLu-177—
[225Ac]Ac-SibuDABAc-225Clinical research
[177Lu]Lu-PSMA-617-treatedLu-177Clinical research
[177Lu]Lu-LNC1011Lu-177Clinical research
[211At]At-astatinatedAt-211—
[177Lu]Lu-EB-PSMA-617Lu-177Clinical research
[177Lu]Lu-vipivotideLu-177Approved
[225Ac]Ac-225-DOTA-J591Ac-225Clinical research

Other entries

AgentIsotopeStageRuns
[225Ac]Ac-PSMA-RLTAc-225—

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