By indication / Neuroendocrine neoplasms

Neuroendocrine neoplasms

20 imaging agents and 35 therapeutic agents reported for this indication. Stage reflects how far each has been taken, not what is available in any given country.

Imaging

AgentIsotopeStageRuns
[68Ga]Ga-DOTA-TOC
paired with [177Lu]Lu-DOTA-TOC
Ga-68Approved40
[18F]FDOPAF-18Approved26
[68Ga]Ga-DOTATATE
paired with [177Lu]Lu-DOTATATE
Ga-68Approved26
[18F]SiTATEF-18—6
[68Ga]Ga-DOTANOC
paired with [47Sc]Sc-DOTANOC
Ga-68—6
[18F]FETrpF-18Research5
[18F]AmBF3-TATEF-18Preclinical3
[18F]AlF-NOTA-octreotideF-18—2
[68Ga]Ga-DOTA-CP04Ga-68—2
[64Cu]Cu-sartate
paired with [67Cu]Cu-SARTATE
Cu-64Clinical research1
[18F]FB(ePEG12)12-exendin-4F-18Clinical research1
[123I]MIBG
paired with [131I]MIBG
I-123—1
[68Ga]TATE-46Ga-68Preclinical1
[203Pb]eSOMA-01Pb-203Reported once1
[203Pb]eSOMA-02Pb-203Reported once1
[203Pb]eSOMA-03Pb-203Reported once1
[68Ga]C803-GIPGa-68Reported once1
[64Cu]Cu-DOTATATE
paired with [177Lu]Lu-DOTATATE
Cu-64Approved
[18F]FET-bAG-TOCA
paired with [177Lu]Lu-DOTATATE
F-18Research
[68Ga]Ga-DOTA-D-Phe-Tyr3-octreotideGa-68Clinical research

Therapy

AgentIsotopeStageRuns
[177Lu]Lu-DOTA-TOC
paired with [68Ga]Ga-DOTA-TOC
Lu-177—11
[177Lu]Lu-DOTATATE
paired with [68Ga]Ga-DOTATATE
Lu-177Approved10
[212Pb]Pb-PSC-PEG2-TOCPb-212—6
[90Y]Y-DOTA-TOC
paired with [68Ga]Ga-DOTA-TOC
Y-90—6
[177Lu]Lu-DOTA-LM3Lu-177Clinical research6
[211At]At-MABGAt-211Preclinical6
[177Lu]Lu-CP04Lu-177—4
[225Ac]Ac-DOTATATE
paired with [68Ga]Ga-DOTATATE
Ac-225Clinical research4
[161Tb]Tb-DOTATATE
paired with [68Ga]Ga-DOTATATE
Tb-161Preclinical3
[177Lu]Lu-DOTA-JR11Lu-177Clinical research3
[212Pb]Pb-DOTAMTATEPb-212Preclinical3
[90Y]Y-DOTATATE
paired with [68Ga]Ga-DOTATATE
Y-90—2
[161Tb]Tb-DOTA-TOC
paired with [68Ga]Ga-DOTA-TOC
Tb-161Preclinical2
[131I]MIBG
paired with [123I]MIBG
I-131Approved2
[161Tb]Tb-DOTA-LM3Tb-161Clinical research2
[161Tb]Tb-3p-C-NETA
paired with [68Ga]Ga-3p-C-NETA
Tb-161Preclinical1
[225Ac]Ac-DOTA-LM3Ac-225Clinical research1
[90Y]Y-90-DOTATOC/DOTATATEY-90Clinical research1
[177Lu]Lu-DOTA-GA4Lu-177Preclinical1
[177Lu]Lu-DOTA-GA13Lu-177Reported once1
[212Pb]Pb-eSOMA-02Pb-212Reported once1
[153Sm]Sm-DOTATATE
paired with [68Ga]Ga-DOTATATE
Sm-153Preclinical
[225Ac]Ac-DOTA-TOC
paired with [68Ga]Ga-DOTA-TOC
Ac-225Clinical research
[213Bi]Bi-DOTA-TOC
paired with [68Ga]Ga-DOTA-TOC
Bi-213Clinical research
[90Y]Y-DOTA-DPhe1-Tyr3-octreotideY-90—
[177Lu]Lu-oxodotreotideLu-177—
[177Lu]Lu-EB-TATELu-177—
[177Lu]Lu-HA-DOTATATELu-177Clinical research
[225Ac]Ac-crown-TATEAc-225—
[166Ho]Ho-166-PLLAHo-166—
[90Y]Y-DOTA-Phe1-Tyr3-octreotideY-90Clinical research
[90Y]Y-microsphereY-90Approved
[177Lu]Lu-LNC1010Lu-177Clinical research
[177Lu]Lu-177-OPS201Lu-177Preclinical
[177Lu]Lu-DOTA-EB-TATELu-177—

Other entries

AgentIsotopeStageRuns
[111In]In-APH070In-111Preclinical1
[212Pb]Pb-VMT-alpha-NETPb-212Clinical research

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