Tracers / [161Tb]Tb-3p-C-NETA

[161Tb]Tb-3p-C-NETA

Also written as [161Tb]Tb-3p-C-NETA; [Tb-161]Tb-3p-C-NETA
Radionuclide
Tb-161 t½ 9907.2 min
Modality
Therapy
Production route
Stage
Syntheses indexed
1

What it is

Compound class
Somatostatin analogue peptide conjugated to NETA-derived chelator (3p-C-NETA-TATE)
Target / mechanism
Somatostatin receptor targeting via TATE (octreotate) peptide PMID 35966589
Clinical application
Theranostic pair
<a href="/tracers/ga68-3pcneta/">ga68-3pcneta</a>

Regulatory status

FDA
EMA (centralised)
Other approvals
Brand names

Clinical use

Typical injected activity
Uptake time

Reported in the literature. Not a dosing recommendation.

Published syntheses

ModuleCassettePurificationYield %RCP %Precursor / supplierSource
Manual synthesisSPE>95%3p-C-NETA35966589
2022 Theranostics
3p-C-NETA was labeled by adding... [161Tb]TbCl3: (4 MBq, 0.1M NaOAc, pH 4.1)... to the 3p-C-NETA solution... and the reaction mixture (V= 1 mL) was incubated for 12 min at the desired temperature. — a RCC of >95% was observed at 40 °C for 3p-C-NETA (10 µM)

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Quality control Preliminary — inferred from compound class

Ph. Eur. monograph
USP monograph
AppearancepHRCP HPLCHPLC UVRadionuclidic (HPGe)Half-lifeActivityEndotoxins (LAL)SterilityFilter integrityOsmolalityMolar activityMetal impurities
How this set was arrived at. base set per Ph. Eur. general monograph 0125 (rule); radiometal tracer -> metal impurities (rule); therapeutic radiopharmaceutical -> osmolality (rule); receptor ligand with a saturable target -> molar activity (rule)

Tests listed by reference only. Monograph texts are copyrighted and are not reproduced here. How these are derived

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Notes

Added from reverse module search (stage 6); 2 article(s) with Tb-161.