Peptide receptor radionuclide therapy

By indication / Peptide receptor radionuclide therapy

2 imaging agents and 32 therapeutic agents reported for this indication. Stage reflects how far each has been taken, not what is available in any given country.

Imaging

Agent	Isotope	Stage	Runs
[68Ga]Ga-DOTATATE paired with [177Lu]Lu-DOTATATE	Ga-68	Approved	26
[64Cu]Cu-sartate paired with [67Cu]Cu-SARTATE	Cu-64	Clinical research	1

Therapy

Agent	Isotope	Stage	Runs
[177Lu]Lu-DOTA-TOC paired with [68Ga]Ga-DOTA-TOC	Lu-177	—	11
[177Lu]Lu-DOTATATE paired with [68Ga]Ga-DOTATATE	Lu-177	Approved	10
[177Lu]Lu-DOTA-MGS5	Lu-177	Clinical research	8
[212Pb]Pb-PSC-PEG2-TOC	Pb-212	—	6
[90Y]Y-DOTA-TOC paired with [68Ga]Ga-DOTA-TOC	Y-90	—	6
[177Lu]Lu-DOTA-LM3	Lu-177	Clinical research	6
[177Lu]Lu-CP04	Lu-177	—	4
[225Ac]Ac-DOTATATE paired with [68Ga]Ga-DOTATATE	Ac-225	Clinical research	4
[161Tb]Tb-DOTATATE paired with [68Ga]Ga-DOTATATE	Tb-161	Preclinical	3
[177Lu]Lu-DOTA-JR11	Lu-177	Clinical research	3
[177Lu]Lu-AMTG	Lu-177	Clinical research	3
[212Pb]Pb-DOTAMTATE	Pb-212	Preclinical	3
[177Lu]Lu-DOTA-PP-F11N	Lu-177	Clinical research	2
[90Y]Y-DOTATATE paired with [68Ga]Ga-DOTATATE	Y-90	—	2
[161Tb]Tb-DOTA-TOC paired with [68Ga]Ga-DOTA-TOC	Tb-161	Preclinical	2
[161Tb]Tb-DOTA-LM3	Tb-161	Clinical research	2
[177Lu]Lu-DOTA-CCK-66 paired with [68Ga]Ga-DOTA-CCK-66	Lu-177	Preclinical	2
[161Tb]Tb-3p-C-NETA paired with [68Ga]Ga-3p-C-NETA	Tb-161	Preclinical	1
[225Ac]Ac-DOTA-LM3	Ac-225	Clinical research	1
[90Y]Y-90-DOTATOC/DOTATATE	Y-90	Clinical research	1
[212Pb]Pb-DOTAM-GRPR1	Pb-212	Preclinical	1
[153Sm]Sm-DOTATATE paired with [68Ga]Ga-DOTATATE	Sm-153	Preclinical
[225Ac]Ac-DOTA-TOC paired with [68Ga]Ga-DOTA-TOC	Ac-225	Clinical research
[213Bi]Bi-DOTA-TOC paired with [68Ga]Ga-DOTA-TOC	Bi-213	Clinical research
[90Y]Y-DOTA-DPhe1-Tyr3-octreotide	Y-90	—
[177Lu]Lu-oxodotreotide	Lu-177	—
[177Lu]Lu-EB-TATE	Lu-177	—
[177Lu]Lu-HA-DOTATATE	Lu-177	Clinical research
[90Y]Y-DOTA-Phe1-Tyr3-octreotide	Y-90	Clinical research
[177Lu]Lu-LNC1010	Lu-177	Clinical research
[177Lu]Lu-177-OPS201	Lu-177	Preclinical
[177Lu]Lu-DOTA-EB-TATE	Lu-177	—

Other entries

Agent	Isotope	Stage	Runs
[111In]In-APH070	In-111	Preclinical	1
[177Lu]Lu-DOTA-cyclo-MG1	Lu-177	Preclinical	1
[177Lu]Lu-DOTA-cyclo-MG2	Lu-177	Preclinical	1
[177Lu]Lu-pentetreotide	Lu-177	Clinical research
[212Pb]Pb-VMT-alpha-NET	Pb-212	Clinical research

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