Tracers / [67Cu]Cu-SARTATE

[67Cu]Cu-SARTATE

Also written as [Cu-67]Cu-SARTATE; SarTATE
Radionuclide
Cu-67 t½ 3708 min
Modality
Therapy
Production route
Stage
preclinical study
Syntheses indexed
2

What it is

Compound class
CB-TE1A1P-PEG4-LLP2A (VLA-4-targeting peptidomimetic conjugated to CB-TE1A1P chelator)
Target / mechanism
VLA-4 (integrin α4β1) PMID 39911068
Clinical application
Theranostic pair
<a href="/tracers/cu64-sartate/">cu64-sartate</a>

Regulatory status

FDA
EMA (centralised)
Other approvals
Brand names

Clinical use

Typical injected activity
Uptake time

Reported in the literature. Not a dosing recommendation.

Published syntheses

ModuleCassettePurificationYield %RCP %Precursor / supplierSource
Manual synthesis41754861
2026 Pharmaceuticals (Basel)
[67Cu]Cu-SAR-TATE
32414949
2020 J Nucl Med

Need this precursor?We can point you to suppliers for [67Cu]Cu-SARTATE, or handle the enquiry for you.

Get in touch

Notes

Added at stage 21 from therapy-discovered.xlsx (bulk PubMed search by isotope/therapy-type/known-agent, not individually researched yet) -- 1 articles found. Target/mechanism, clinical application, indications, approval and precursor fields still need per-agent research and are intentionally left empty. Diagnostic pair signal at discovery: YES - Cu-64. Compound class inferred from precursor name (not stated outright) -- PMID 39911068: 'CB-TE1A1P-PEG4-LLP2A (LLP2A) was kindly provided by AusPep (34).'. Stage set/updated at stage 23 from PMID 39911068: 'We used orthotopic syngeneic (i.e., B16-F10, B78, 4T1, GL261, TH-MYCN, and E2A-PBX1) and human (i.e., SK-MEL-37, 143B, and IMR-5) cancer models for in vivo PET/CT imaging and biodistribution studies.'.