By indication / Fibroblast activation / tumour stroma

Fibroblast activation / tumour stroma

14 imaging agents and 22 therapeutic agents reported for this indication. Stage reflects how far each has been taken, not what is available in any given country.

Imaging

AgentIsotopeStageSyntheses
[68Ga]Ga-FAPI-46
paired with [177Lu]Lu-FAPI-46
Ga-68Clinical research77
[68Ga]Ga-FAPI-04
paired with [177Lu]Lu-FAPI-04
Ga-6847
[68Ga]Ga-FAPI
paired with [177Lu]Lu-FAPI
Ga-68pilot clinical study25
[18F]FAPI-74F-1811
[18F]AlF-FAPI-74F-1810
[18F]AlF-NOTA-FAPI-04F-187
[68Ga]Ga-OncoFAP-DOTAGAGa-68Research4
[18F]AlF-OncoFAP-NODAGAF-18Research
[18F]AlF-OncoFAP-NOTAF-18Research
[68Ga]Ga-OncoFAP-NODAGAGa-68Research
[68Ga]Ga-OncoFAP-NOTAGa-68Research
[18F]AlF-OncoFAPF-18
[18F]FB-4AH29F-18preclinical
[68Ga]Ga-FAPI-02Ga-68

Therapy

AgentIsotopeStageSyntheses
[177Lu]Lu-FAPI-2286
paired with [64Cu]Cu-FAPI-2286
Lu-1779
[225Ac]Ac-DOTA-4AH29Ac-2252
[212Pb]Pb-FAPI-46
paired with [68Ga]Ga-FAPI-46
Pb-2121
[225Ac]Ac-FAPI-04
paired with [68Ga]Ga-FAPI-04
Ac-225preclinical1
[177Lu]Lu-DOTA-2P(FAPI)2Lu-177preclinical1
[177Lu]Lu-DOTA-NI-FAPI-04Lu-177preclinical1
[68Ga]PEG2-COUGa-68Reported once1
[68Ga]PEG6-COUGa-68Reported once1
[177Lu]Lu-CHX-A''-DTPA-F8Lu-177Reported once1
[89Zr]Nb159Zr-89Reported once1
[89Zr]PEG-Nb159Zr-89Reported once1
[177Lu]Lu-PEG-Nb159
paired with [89Zr]PEG-Nb159
Lu-177preclinical study1
[111In]DOTAGA-FAP-2286In-111Reported once1
[225Ac]Ac-DOTAGA-FAP-2286-ALBAc-225Reported once1
[18F]AlF-H3RESCA-FAPIF-18preclinical study1
[225Ac]Ac-DOTA-PKU525Ac-225Reported once1
[177Lu]Lu-DOTA-PEG7-tetrazineLu-177preclinical study1
[111In]eFAP-6
paired with [177Lu]Lu-eFAP-6
In-111Reported once1
[177Lu]Lu-eFAP-6
paired with [111In]eFAP-6
Lu-177preclinical study1
[68Ga]DOTA-FD1
paired with [177Lu]Lu-DOTA-FD1
Ga-68Reported once1
[68Ga]DOTA-FD2
paired with [177Lu]Lu-DOTA-FD2
Ga-68Reported once1
[68Ga]SB02055Ga-68preclinical study1

Have a question?Reagents, modules, introductions to manufacturers or to specialists in your region — tell us what you need.

Get in touch