By indication / Other radioligand therapy

Other radioligand therapy

4 imaging agents and 22 therapeutic agents reported for this indication. Stage reflects how far each has been taken, not what is available in any given country.

Imaging

AgentIsotopeStageRuns
[18F]FBPAF-18Preclinical6
[99mTc]Tc-PSMA-I&STc-99m—4
[89Zr]Zr-DFO-girentuximabZr-89Clinical research1
[18F]fluorophenylalanineF-18Clinical research

Therapy

AgentIsotopeStageRuns
[225Ac]Ac-DOTA-YS5Ac-225Preclinical4
[177Lu]Lu-pentixatherLu-177Clinical research3
[177Lu]Lu-PP-F11NLu-177Clinical research3
[225Ac]Ac-Macropa-PEG4-YS5Ac-225—3
[131I]MIBG
paired with [123I]MIBG
I-131Approved2
[177Lu]Lu-AKIR001Lu-177Clinical research2
[177Lu]Lu-DOTA-DV1-K-DV3Lu-177Preclinical2
[225Ac]Ac-DOTA-CCK-66Ac-225Preclinical1
[225Ac]Ac-DOTAZOLAc-225Preclinical1
[131I]I-131-PD-L1I-131—1
[90Y]Y-90-FF-21101Y-90Clinical research1
[161Tb]Tb-BL02Tb-161Preclinical1
[225Ac]Ac-mcp-TDI-Y-010Ac-225Reported once1
[177Lu]Lu-DOTA-GA13Lu-177Reported once1
[161Tb]Tb-cAC10Tb-161Reported once1
[225Ac]Ac(MacropaSq-hG250)Ac-225Preclinical1
[177Lu]Lu-DTPA-NY003Lu-177Preclinical1
[90Y]Y-pentixatherY-90—
[211At]At-211-AMT
paired with [11C]AMT
At-211Preclinical
[177Lu]Lu-CE-21
paired with [68Ga]CE-21
Lu-177Clinical research
[212Pb]Pb-DO3A-PEG7-TzPb-212Preclinical
2-[211At]astato-α-methyl-L-phenylalanineAt-211Preclinical

Other entries

AgentIsotopeStageRuns
[111In]In-minigastrinIn-111—2
[177Lu]Lu-DOTA-A1K2Lu-177Preclinical1
[177Lu]Lu-DOTA-M5ALu-177Preclinical1
[90Y]Y-DOTA-ARY-90Preclinical1
[188Re]Re-Tin colloidRe-188—1
[166Ho]Ho-DTPAHo-166Preclinical
[161Tb]Tb-DOTA-IBATb-161Clinical research
[213Bi]Bi-B-B4Bi-213Preclinical
[211At]At-(RGD)4At-211Preclinical
[177Lu]Lu-hydroxyapatiteLu-177Preclinical
[166Ho]Ho-labeled microspheresHo-166Preclinical
[153Sm]Sm-HASm-153Approved
[211At]At-antiCD33At-211Preclinical
[188Re]Re-6D2Re-188Clinical research
[212Pb]Pb-DOTA-Re(Arg11)CCMSHPb-212Preclinical

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