Tracers / [177Lu]Lu-DOTA-TRK-950

[177Lu]Lu-DOTA-TRK-950

Also written as [Lu-177]Lu-DOTA-TRK-950
Radionuclide
Lu-177 t½ 9584.6 min
Modality
Therapy
Production route
Stage
Reported once
Syntheses indexed
1

What it is

Compound class
DOTA-conjugated anti-CAPRIN-1 monoclonal antibody (radioimmunoconjugate)
Target / mechanism
Targets CAPRIN-1, a cancer-specific cell surface antigen PMID 40473914
Clinical application
Theranostic pair
<a href="/tracers/in111-dotatrk950/">in111-dotatrk950</a>

Regulatory status

FDA
EMA (centralised)
Other approvals
Brand names

Clinical use

Typical injected activity
Uptake time

Reported in the literature. Not a dosing recommendation.

Published syntheses

ModuleCassettePurificationYield %RCP %Precursor / supplierSource
Manual synthesis≥ 95%TRK-950-DOTA
ITM
40473914
2025 J Cancer Res Clin Oncol
Radiolabeling with 177Lu was performed using a modified version of the above method.

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Notes

Added at stage 22: promoted from 'Reported once' (single-article, no diagnostic pair at discovery) because a full-text synthesis with extracted data exists in parsed-therapy.xlsx -- PMID(s): 40473914. Target/mechanism, clinical application, indications, approval and precursor fields still need per-agent research and are intentionally left empty. Compound class inferred from precursor name (not stated outright) -- PMID 40473914: 'TRK-950-DOTA'.