Tracers / [18F]FBnTP

[18F]FBnTP

Also written as [18F]FBnTP; [F-18]FBnTP
Radionuclide
F-18 t½ 109.77 min
Modality
PET
Production route
Stage
Syntheses indexed
2

What it is

Compound class
lipophilic phosphonium cation (triphenylphosphonium derivative)
Target / mechanism
Mitochondrial membrane potential sensor; cellular uptake correlated with mitochondrial oxidative phosphorylation PMID 38935218
Clinical application
Imaging of myocardial perfusion, coronary artery stenosis severity, ischemic area delineation, apoptosis detection/quantification, and oncological diagnosis and therapeutic monitoring PMID 38935218
Theranostic pair

Regulatory status

FDA
EMA (centralised)
Other approvals
Brand names

Clinical use

Typical injected activity
Uptake time

Reported in the literature. Not a dosing recommendation.

Published syntheses

ModuleCassettePurificationYield %RCP %Precursor / supplierSource
ELIXYS FLEX/CHEM
Sofie Biosciences
vendor cassetteSPE28.6 ± 5.1 %
yes
> 99 %4-trimethylammoniumbenzaldehyde trifluoromethanesulfonate
ABX
28905308
2018 Mol Imaging Biol
a three-pot, four-step synthesis was implemented on the ELIXYS FLEX/CHEM radiosynthesizer (Sofie Biosciences) — RCY = 28.6 ± 5.1 % with n = 3
TRACERlab FX FN
GE HealthCare
custom manifoldHPLC+SPE28.33 ± 13.92%
no
99.79 ± 0.41%triphenyl(4‐(4,4,5,5‐tetramethyl‐1,3,2‐dioxaborolan‐2‐yl)benzyl)phosphonium trifluoromethanesulfonate
MilliporeSigma
38935218
2024 EJNMMI Radiopharm Chem
GE TRACERlab™ FXFN, the most widely used synthesis module for routine clinical radiopharmaceutical production — radiochemical yields ranging from 28.33 ± 13.92% (non-decay corrected)

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Quality control Preliminary — inferred from compound class

Ph. Eur. monograph
USP monograph
AppearancepHRCP HPLCRCP TLCHPLC UVRadionuclidic (HPGe)Half-lifeActivityEndotoxins (LAL)SterilityFilter integrity
How this set was arrived at. base set per Ph. Eur. general monograph 0125 (rule); organic-phase radiosynthesis assumed from isotope/compound class, no synthesis data confirming it -> GC residual solvents (preliminary); conventional nucleophilic 18F-fluorination assumed from isotope/compound class, no synthesis data confirming K222 use -> Kryptofix test (preliminary)

Tests listed by reference only. Monograph texts are copyrighted and are not reproduced here. How these are derived

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Notes

Added from reverse module search (stage 6); 2 article(s) with F-18.