Tracers / [11C]DASB

[11C]DASB

Also written as [11C]DASB; [C-11]DASB; DASB
Radionuclide
C-11 t½ 20.36 min
Modality
PET
Production route
Stage
Syntheses indexed
4

What it is

Compound class
O-desmethyl DASB derived carbon-11 methylated arylthiophenylamine SERT ligand
Target / mechanism
Serotonin transporter (SERT) PMID 36071112
Clinical application
Theranostic pair

Regulatory status

FDA
EMA (centralised)
Other approvals
Brand names

Clinical use

Typical injected activity
Uptake time

Reported in the literature. Not a dosing recommendation.

Published syntheses

ModuleCassettePurificationYield %RCP %Precursor / supplierSource
TRACERlab FX C Pro
GE HealthCare
custom manifoldHPLC+SPE3.0%
no
>95%O-desmethyl DASB
ABX
23123138
2013 Nucl Med Biol
Ethanolic loop chemistry is fully automated using a GE TRACERLab FXC-Pro synthesis module — 3.0% RCY; >95% RCP; SA = 15152 Ci/mmol; n = 9
TRACERlab FX C Pro
GE HealthCare
custom manifoldHPLC+SPE3.0%
no
>95%O-desmethyl DASB
ABX
23123138
2013 Nucl Med Biol
Ethanolic loop chemistry is fully automated using a GE TRACERLab FXC-Pro synthesis module — 3.0% RCY; >95% RCP; SA = 10931 Ci/mmol; n = 3
36071112
2022 Mol Psychiatry
66.3+/-6.9%
yes
[11C]CH3I19359188
2009 Appl Radiat Isot

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Quality control Preliminary — inferred from compound class

Ph. Eur. monograph
USP monograph
AppearancepHRCP HPLCRCP TLCHPLC UVRadionuclidic (HPGe)Half-lifeActivityEndotoxins (LAL)SterilityFilter integrity
How this set was arrived at. base set per Ph. Eur. general monograph 0125 (rule); organic-phase radiosynthesis assumed from isotope/compound class, no synthesis data confirming it -> GC residual solvents (preliminary)

Tests listed by reference only. Monograph texts are copyrighted and are not reproduced here. How these are derived

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Notes

Added from reverse module search (stage 6); 2 article(s) with C-11. Compound class inferred from precursor name (not stated outright) -- PMID 23123138: 'O-desmethyl DASB (1.0 mg) in ethanol (100 µL)'.